SCHEMBL7410149

SCHEMBL7410149

C=C(COc1ccc(Br)cc1)C(=O)OC

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
KDM4E B2RXH2 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
MAPT P10636 2/20 0.48
POLB P06746 2/20 0.46
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
TP53 P04637 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410091 0.84 MAPT (0.49) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL11035215 0.83 GAA (0.51) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL11076225 0.83 ALOX15 (0.55) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL12451865 0.83 ALDH1A1 (0.53) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL4115419 0.79 PTGS2 (0.57) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL13403114 0.77 ALDH1A1 (0.64) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL8215730 0.76 L3MBTL1 (0.51) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL31110815 0.75 KMT2A (0.38) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL28079414 0.75 GSK3B (0.48) ALDH1A1MEN1KMT2AMAPTPOLB
SCHEMBL13382671 0.74 POLB (0.54) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939418-A ANTICOAGULANT THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1999-08-17 US disclosed
EP-0874629-A4 ISOXAZOLINE, ISOTHIAZOLINE AND PYRAZOLINE FACTOR Xa INHIBITORS DU PONT MERCK PHARMA (US) 1999-08-04 EP disclosed
EP-0874629-A1 ISOXAZOLINE, ISOTHIAZOLINE AND PYRAZOLINE FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-11-04 EP disclosed
WO-1997023212-A1 ISOXAZOLINE, ISOTHIAZOLINE AND PYRAZOLINE FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-07-03 WO disclosed