SCHEMBL7410932

SCHEMBL7410932

CC(=O)SCC(C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O)C(F)(F)F

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ACE P12821 4/20 0.61
ALOX15 P16050 1/20 0.60
ECE1 P42892 9/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11430738 0.87 ACE (0.67) ACEALOX15ECE1
SCHEMBL7322267 0.86 ACE (0.73) ACEALOX15ECE1
SCHEMBL7410432 0.85 ACE (0.71) ACEECE1
SCHEMBL7419934 0.84 MME (0.53) ACEECE1
SCHEMBL6172199 0.83 LTA4H (0.69) ACEALOX15ECE1
SCHEMBL6172205 0.83 LTA4H (0.69) ACEALOX15ECE1
SCHEMBL9068531 0.82 ECE1 (0.75) ACEALOX15ECE1
SCHEMBL7416436 0.81 MME (0.51) ACEECE1
SCHEMBL7411840 0.81 MMP1 (0.43) ACEALOX15
SCHEMBL7411850 0.81 MMP1 (0.43) ACEALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5414013-A Enzyme inhibitors E. R. SQUIBB & SONS, INC. (US) 1995-05-09 US disclosed
US-5414017-A Cardiovascular agents E. R. SQUIBB & SONS, INC. (US) 1995-05-09 US disclosed
EP-0449523-B1 Mercapto- or acylthio-trifluoromethyl amide derivatives and their use SQUIBB & SONS INC (US) 1994-08-17 EP disclosed
US-5223516-A Endopeptidase inhibitors E. R. SQUIBB & SONS, INC. (US) 1993-06-29 US disclosed
EP-0449523-A1 Mercapto- or acylthio-trifluoromethyl amide derivatives and their use E.R. SQUIBB & SONS, INC. (US) 1991-10-02 EP disclosed