SCHEMBL7410984

SCHEMBL7410984

N[C@@H](CCc1c(O)noc1-c1cccs1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.39
RORC P51449 1/20 0.37
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
ALDH1A1 P00352 3/20 0.36
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
CYP2C19 P33261 2/20 0.35
GRM6 O15303 2/20 0.34
ALOX15 P16050 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
SLC1A3 P43003 1/20 0.34
SLC1A2 P43004 1/20 0.34
SLC1A1 P43005 1/20 0.34
DAGLA Q9Y4D2 1/20 0.34
MAPT P10636 2/20 0.34
HSD17B10 Q99714 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7372989 1.00 MCL1 (0.39) MCL1RORCMEN1KMT2AALDH1A1
SCHEMBL7049750 0.88 GRIA1 (0.40) MCL1RORCNPC1RAB9ANPSR1
SCHEMBL7371185 0.88 GRIA1 (0.40) MCL1RORCNPC1RAB9ANPSR1
SCHEMBL8128585 0.81 KIF11 (0.39) MEN1KMT2ACYP2C19GRM6ALOX15
SCHEMBL8128581 0.81 KIF11 (0.39) MEN1KMT2ACYP2C19GRM6ALOX15
SCHEMBL7452730 0.80 SLC1A3 (0.35) MEN1KMT2ACYP2C19GRM6ALOX15
SCHEMBL7452720 0.80 SLC1A3 (0.35) MEN1KMT2ACYP2C19GRM6ALOX15
SCHEMBL7365968 0.79 TAAR1 (0.42) MCL1RORCMEN1KMT2ANPC1
SCHEMBL8119688 0.77 GRIA1 (0.53) MCL1RORCMEN1KMT2ACYP2C19
SCHEMBL8119682 0.77 GRIA1 (0.53) MCL1RORCMEN1KMT2ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994107-A1 5-Arylisoxazol-4-yl-substituted 2-amino carboxylic acid compounds H. LUNDBECK A/S (DK) 2000-04-19 EP disclosed
EP-0726896-A1 5-ARYLISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1996-08-21 EP disclosed
WO-1995012587-A1 5-ARYLISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1995-05-11 WO disclosed