SCHEMBL8128581

SCHEMBL8128581

NC(CCc1c(O)noc1-c1ccccc1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.39
PTPN1 P18031 1/20 0.39
GRM6 O15303 2/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
ALPI P09923 1/20 0.37
PKM P14618 1/20 0.37
PTGS1 P23219 1/20 0.37
XIAP P98170 1/20 0.37
SLC7A5 Q01650 1/20 0.37
NOS1 P29475 1/20 0.36
SLC7A11 Q9UPY5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8128585 1.00 KIF11 (0.39) KIF11PTPN1GRM6MEN1CYP1A2
SCHEMBL8125242 0.92 NOS1 (0.43) KIF11PTPN1KMT2ANOS1
SCHEMBL8125246 0.92 NOS1 (0.43) KIF11PTPN1KMT2ANOS1
SCHEMBL7406141 0.88 TPH1 (0.46) KIF11GRM6MEN1CYP1A2CYP2C9
SCHEMBL7406145 0.88 TPH1 (0.46) KIF11GRM6MEN1CYP1A2CYP2C9
SCHEMBL7408342 0.87 SLC7A11 (0.45) KIF11MEN1CYP1A2KMT2ASLC7A11
SCHEMBL7408347 0.87 SLC7A11 (0.45) KIF11MEN1CYP1A2KMT2ASLC7A11
SCHEMBL7159040 0.86 SLC7A5 (0.46) PTPN1ALPIPKMPTGS1XIAP
SCHEMBL8129370 0.86 SLC7A5 (0.46) PTPN1ALPIPKMPTGS1XIAP
SCHEMBL7159035 0.86 SLC7A5 (0.46) PTPN1ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1056837-C 5-arylisoxazol-4-yl-substituted 2-aminocarboxylic acid compounds LUNDBECK & CO AS H (DK) 2000-09-27 CN disclosed
EP-0994107-A1 5-Arylisoxazol-4-yl-substituted 2-amino carboxylic acid compounds H. LUNDBECK A/S (DK) 2000-04-19 EP disclosed
CN-1136810-A 5-arylisoxazol-4-yl-substituted 2-aminocarboxylic acid compounds LUNDBECK & CO AS H (DK) 1996-11-27 CN disclosed