SCHEMBL7410985

SCHEMBL7410985

O=S(=O)(Cc1ccccc1)C1=NC=C[N]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
FAAH O00519 1/20 0.44
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
ELANE P08246 1/20 0.44
PRTN3 P24158 1/20 0.44
PRSS3 P35030 1/20 0.44
CA5A P35218 1/20 0.44
CA9 Q16790 1/20 0.44
ALDH1A1 P00352 4/20 0.42
MAPT P10636 4/20 0.42
HPGD P15428 3/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
AKR1B1 P15121 1/20 0.42
TSHR P16473 3/20 0.42
HSD17B10 Q99714 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
POLB P06746 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzylsulfonylbenzene SCHEMBL780337 0.69 TSHR (0.68) CA1CA2FAAHPRSS1PRSS2
Benzylsulfonylbenzene SCHEMBL1877584 0.67 TSHR (0.66) CA1CA2FAAHPRSS1PRSS2
SCHEMBL10728701 0.67 ALDH1A1 (0.50) CA1CA2FAAHPRSS1PRSS2
SCHEMBL8887464 0.67 TSHR (0.42) CA1CA2FAAHPRSS1PRSS2
SCHEMBL2233216 0.66 CA2 (0.58) CA1CA2FAAHPRSS1PRSS2
SCHEMBL3626579 0.66 CA2 (0.52) CA1CA2FAAHPRSS1PRSS2
SCHEMBL29482080 0.65 TSHR (0.58) CA1CA2FAAHPRSS1PRSS2
SCHEMBL9870797 0.65 KMT2A (0.51) CA1CA2FAAHPRSS1PRSS2
SCHEMBL88641 0.65 CA2 (0.64) CA1CA2FAAHPRSS1PRSS2
SCHEMBL2767017 0.64 ALDH1A1 (0.56) CA1CA2FAAHPRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946508-A1 NITROGEN CONTAINING HETEROAROMATICS AS FACTOR Xa INHIBITORS Du Pont Pharmaceuticals Company (US) 1999-10-06 EP disclosed
EP-0946528-A2 OXYGEN OR SULFUR CONTAINING 5-MEMBERED HETEROAROMATICS AS FACTOR Xa INHIBITORS Du Pont Pharmaceuticals Company (US) 1999-10-06 EP disclosed
WO-1998028269-A1 NITROGEN CONTAINING HETEROAROMATICS AS FACTOR Xa INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 1998-07-02 WO disclosed
WO-1998028282-A2 OXYGEN OR SULFUR CONTAINING 5-MEMBERED HETEROAROMATICS AS FACTOR Xa INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 1998-07-02 WO disclosed