SCHEMBL7411767

SCHEMBL7411767

Fc1ccc(CNC(c2ccc(F)cc2)C2CCN(CCc3ccccc3)CC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.59
HTR2C P28335 2/20 0.59
HTR7 P34969 1/20 0.59
KDM4E B2RXH2 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
TSHR P16473 1/20 0.52
SLC6A4 P31645 1/20 0.52
SLC6A3 Q01959 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9330147 0.79 HTR2A (0.87) HTR2AHTR2CHTR7KDM4ECYP1A2
SCHEMBL28781802 0.78 ACHE (0.76) SLC6A4SLC6A3
SCHEMBL7417986 0.77 PKM (0.51)
SCHEMBL7409826 0.77 ALDH1A1 (0.46) HTR2AHTR2CHTR7TSHR
SCHEMBL9328582 0.77 HTR2A (0.87) HTR2AHTR2CHTR7KDM4ECYP1A2
Hydrochloric Acid SCHEMBL7411439 0.76 HTR2A (0.67) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL1505925 0.76 SLC6A4 (0.61) CYP2D6SLC6A4SLC6A3
SCHEMBL7416706 0.75 KMT2A (0.47) HTR2ATSHR
SCHEMBL7219033 0.74 HRH3 (0.51)
SCHEMBL7417922 0.73 RPS6KB1 (0.43) HTR2ASLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5198449-A N-substituted alpha-arylazacycloalkylmethanamines and their use as cardiovascular agents A. H. ROBINS COMPANY INCORPORATED (US) 1993-03-30 US disclosed