SCHEMBL7413028

SCHEMBL7413028

CNC(=O)N(Cc1ccc(F)cc1)C(c1ccc(F)cc1)C1CCN(CCc2ccccc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.57
TMEM97 Q5BJF2 2/20 0.57
HTR2A P28223 2/20 0.52
HTR2C P28335 1/20 0.52
HTR7 P34969 1/20 0.52
CACNA1G O43497 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416616 0.89 OPRM1 (0.60) OPRM1TMEM97HTR2AHTR2CHTR7
SCHEMBL7412596 0.86 HTR2A (0.41) OPRM1TMEM97HTR2AHTR2CHTR7
SCHEMBL7409872 0.84 HTR2A (0.43) OPRM1TMEM97HTR2ACACNA1G
SCHEMBL7419477 0.76 HTR2A (0.48) OPRM1TMEM97HTR2A
SCHEMBL9330147 0.73 HTR2A (0.87) HTR2AHTR2CHTR7
SCHEMBL28781746 0.73 OPRM1 (1.00) OPRM1TMEM97
SCHEMBL28781770 0.72 OPRM1 (0.80) OPRM1TMEM97
SCHEMBL7416706 0.71 KMT2A (0.47) OPRM1TMEM97HTR2A
SCHEMBL28781760 0.71 OPRM1 (1.00) OPRM1TMEM97
SCHEMBL9328582 0.71 HTR2A (0.87) TMEM97HTR2AHTR2CHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5198449-A N-substituted alpha-arylazacycloalkylmethanamines and their use as cardiovascular agents A. H. ROBINS COMPANY INCORPORATED (US) 1993-03-30 US disclosed