SCHEMBL7413329

SCHEMBL7413329

C[C@@H]1OCC(=O)[C@H]1NC(=O)[CH]C[C@@](C)(Cc1ccccc1)C(N)=O

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
MME P08473 1/20 0.32
ACE P12821 1/20 0.32
NAAA Q02083 2/20 0.32
CYP1A2 P05177 1/20 0.31
RECQL P46063 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590297 1.00 CYP3A4 (0.34) CYP3A4ALDH1A1CYP2C9CYP2C19MME
SCHEMBL6588900 0.90 NAAA (0.35) NAAA
SCHEMBL7412446 0.90 NAAA (0.35) NAAA
SCHEMBL6589398 0.89 CTSL (0.38) CYP3A4ALDH1A1CYP2C9CYP2C19NAAA
SCHEMBL7420898 0.89 CTSL (0.38) CYP3A4ALDH1A1CYP2C9CYP2C19NAAA
SCHEMBL7416310 0.84 MAPT (0.33)
SCHEMBL6586616 0.84 MAPT (0.33)
SCHEMBL6586151 0.84 ALDH1A1 (0.31) CYP3A4ALDH1A1CYP2C9CYP2C19
SCHEMBL6590478 0.83 HRH3 (0.34) CYP3A4ALDH1A1CYP2C9CYP2C19MME
SCHEMBL7418471 0.79 CTSL (0.37) NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002544274-A 2002-12-24 JP claimed
EP-1178986-A2 FURANONE DERIVATIVES AS INHIBITORS OF CATHEPSIN S Medivir UK Ltd (GB) 2002-02-13 EP claimed
WO-2000069855-A2 FURANONE DERIVATIVES AS INHIBITORS OF CATHEPSIN S MEDIVIR UK LIMITED (GB) 2000-11-23 WO claimed
EP-1178986-A2 FURANONE DERIVATIVES AS INHIBITORS OF CATHEPSIN S Medivir UK Ltd (GB) 2002-02-13 EP disclosed
WO-2000069855-A2 FURANONE DERIVATIVES AS INHIBITORS OF CATHEPSIN S MEDIVIR UK LIMITED (GB) 2000-11-23 WO disclosed