SCHEMBL7413846

SCHEMBL7413846

C#Cc1ccccc1C(F)(F)Br

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA5A P35218 1/20 0.31
CA9 Q16790 1/20 0.31
PTPN1 P18031 2/20 0.31
AR P10275 1/20 0.31
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
SLC22A12 Q96S37 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL313726 0.83 ALDH1A1 (0.40) ARALDH1A1POLBTDP1L3MBTL1
SCHEMBL4204571 0.76 ALDH1A1 (0.40) CA1CA2CA5ACA9ALDH1A1
SCHEMBL10538304 0.74 KIF11 (0.34) AR
SCHEMBL717061 0.73 ALDH1A1 (0.46) CA2ALDH1A1TDP1
SCHEMBL5051929 0.73 MEN1 (0.30) POLB
SCHEMBL28870 0.73 HDAC8 (0.36) ALDH1A1
SCHEMBL29549283 0.73 HDAC8 (0.36) ALDH1A1
SCHEMBL1117918 0.70 KCNN4 (0.46) CA1CA2CA5ACA9AR
SCHEMBL30185685 0.70 HDAC8 (0.35)
SCHEMBL27884965 0.70 ALDH1A1 (0.33) CA2ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5256677-A Enzyme inhibitor for treating acquired immune deficiency syndrome ABBOTT LABORATORIES (US) 1993-10-26 US disclosed
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO disclosed
US-5151438-A Enzyme inhibitors for treatment of aids ABBOTT LABORATORIES (US) 1992-09-29 US disclosed