SCHEMBL7414248

SCHEMBL7414248

CN1C2CCCC1CC(NC(=O)c1cc(Cl)cc3c1OCCO3)C2

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 8/20 0.52
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HTR4 Q13639 1/20 0.45
KCNH2 Q12809 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416813 0.91 HTR3A (0.52) HTR3AMEN1KMT2AHTR4KCNH2
SCHEMBL7271062 0.84 DRD2 (0.53) HTR3AMEN1KMT2AHTR4KCNH2
SCHEMBL7270659 0.80 DRD2 (0.52) HTR3AMEN1KMT2AHTR4KCNH2
SCHEMBL7302570 0.79 HTR4 (0.61) HTR3AHTR4KCNH2
SCHEMBL7302326 0.79 HTR4 (0.61) HTR3AHTR4KCNH2
Hydrochloric Acid SCHEMBL7377307 0.79 HTR4 (0.61) HTR3AHTR4KCNH2
Hydrochloric Acid SCHEMBL7377304 0.79 HTR4 (0.61) HTR3AHTR4KCNH2
SCHEMBL8939976 0.78 HTR3A (0.49) HTR3AMEN1KMT2AHTR4KCNH2
SCHEMBL7270890 0.77 HTR3A (0.48) HTR3AMEN1KMT2AHTR4KCNH2
SCHEMBL7417950 0.76 HTR3A (0.48) HTR3AMEN1KMT2AHTR4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0561910-A1 PHARMACEUTICALS BEECHAM GROUP PLC (GB) 1993-09-29 EP claimed
WO-1992010494-A1 PHARMACEUTICALS BEECHAM GROUP P.L.C. (GB) 1992-06-25 WO claimed
WO-1992010494-A1 PHARMACEUTICALS BEECHAM GROUP P.L.C. (GB) 1992-06-25 WO disclosed