SCHEMBL7414440

SCHEMBL7414440

CN(C)/C=C/c1cc(CC(=O)O)ccc1[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 6/20 0.44
ALDH1A1 P00352 3/20 0.40
MAPT P10636 2/20 0.40
CYP1A2 P05177 1/20 0.40
SIRT5 Q9NXA8 3/20 0.39
STAT3 P40763 1/20 0.39
PTGS2 P35354 1/20 0.39
GSTP1 P09211 1/20 0.38
GSTM2 P28161 1/20 0.38
PTGS1 P23219 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414442 1.00 BACE1 (0.44) BACE1ALDH1A1MAPTCYP1A2SIRT5
SCHEMBL7411663 0.90 PTGS2 (0.47) BACE1ALDH1A1MAPTCYP1A2STAT3
SCHEMBL7411665 0.90 PTGS2 (0.47) BACE1ALDH1A1MAPTCYP1A2STAT3
SCHEMBL7006042 0.80 CASP6 (0.55) BACE1ALDH1A1MAPT
SCHEMBL7006045 0.80 CASP6 (0.55) BACE1ALDH1A1MAPT
SCHEMBL7006049 0.80 CASP6 (0.55) BACE1ALDH1A1MAPT
SCHEMBL11837128 0.77 ATM (0.50) BACE1ALDH1A1MAPTCYP1A2SIRT5
SCHEMBL11837114 0.77 ATM (0.50) BACE1ALDH1A1MAPTCYP1A2SIRT5
SCHEMBL13778767 0.77 MAPT (0.48) BACE1ALDH1A1MAPTPTGS2AKR1C3
SCHEMBL12367389 0.76 TSHR (0.53) BACE1ALDH1A1MAPTPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380739-A Angiotensin II antagonists SYNTEX (U.S.A.) INC. (US) 1995-01-10 US disclosed
US-5212195-A Substituted indole antagonists derivatives which are angiotensin II SYNTEX (U.S.A.) INC. (US) 1993-05-18 US disclosed