SCHEMBL7414680

SCHEMBL7414680

O=C(c1ccc(C(F)(F)F)cc1)C1CCN(Cc2ccc3ccccc3c2)CC1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 2/20 0.66
MCHR1 Q99705 7/20 0.58
HTR2A P28223 2/20 0.53
ACHE P22303 1/20 0.52
SIGMAR1 Q99720 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7412259 0.87 MCHR1 (0.71) MCHR1HTR2A
SCHEMBL7417801 0.87 MCHR1 (0.68) MCHR1HTR2AACHESIGMAR1
SCHEMBL5539621 0.86 SIGMAR1 (0.65) DRD4HTR2ASIGMAR1
SCHEMBL7412406 0.83 MEN1 (0.66) DRD4MCHR1
SCHEMBL7415439 0.83 MCHR1 (0.72) MCHR1HTR2AACHESIGMAR1
SCHEMBL7304448 0.78 MCHR1 (0.65) MCHR1ACHESIGMAR1
SCHEMBL6210244 0.77 HTR2A (0.69) MCHR1HTR2A
SCHEMBL7410338 0.75 MCHR1 (0.60) MCHR1HTR2A
Trifluoroacetic Acid SCHEMBL1921350 0.74 MCHR1 (0.58) MCHR1ACHESIGMAR1
SCHEMBL24529849 0.74 SIGMAR1 (0.62) ACHESIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5198449-A N-substituted alpha-arylazacycloalkylmethanamines and their use as cardiovascular agents A. H. ROBINS COMPANY INCORPORATED (US) 1993-03-30 US disclosed