SCHEMBL7415439

SCHEMBL7415439

O=C(c1ccc(F)c(F)c1)C1CCN(Cc2ccc3ccccc3c2)CC1

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 8/20 0.72
HTR2A P28223 2/20 0.54
CCR3 P51677 1/20 0.53
ACHE P22303 1/20 0.53
ALDH1A1 P00352 1/20 0.53
SIGMAR1 Q99720 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7412259 0.88 MCHR1 (0.71) MCHR1HTR2ACCR3
SCHEMBL7417801 0.86 MCHR1 (0.68) MCHR1HTR2ACCR3ACHESIGMAR1
SCHEMBL7414680 0.83 DRD4 (0.66) MCHR1HTR2AACHESIGMAR1
SCHEMBL7412406 0.82 MEN1 (0.66) MCHR1CCR3
SCHEMBL6210244 0.81 HTR2A (0.69) MCHR1HTR2ACCR3
SCHEMBL7304448 0.79 MCHR1 (0.65) MCHR1CCR3ACHESIGMAR1
SCHEMBL7413680 0.77 MCHR1 (0.59) MCHR1
SCHEMBL7410338 0.76 MCHR1 (0.60) MCHR1HTR2ACCR3
SCHEMBL4795273 0.74 S1PR5 (0.62) MCHR1CCR3ACHESIGMAR1
SCHEMBL4795270 0.74 S1PR5 (0.62) MCHR1CCR3ACHESIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5198449-A N-substituted alpha-arylazacycloalkylmethanamines and their use as cardiovascular agents A. H. ROBINS COMPANY INCORPORATED (US) 1993-03-30 US disclosed