SCHEMBL7414772

SCHEMBL7414772

CC#CCOc1ccc(SC(CCCCNC(=O)CNC(=O)c2ccc3ccccc3n2)C(=O)NO)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 12/20 0.57
MMP9 P14780 6/20 0.57
MMP13 P45452 6/20 0.57
MAPT P10636 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
MMP1 P03956 3/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
HDAC1 Q13547 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7413633 0.87 ADAM17 (0.56) ADAM17MMP9MMP13MMP1HDAC1
SCHEMBL7415917 0.86 ADAM17 (0.58) ADAM17MMP9MMP13MMP1HDAC1
SCHEMBL7413415 0.84 MAPT (0.39) ADAM17MMP9MMP13MAPTL3MBTL1
SCHEMBL3939996 0.82 ADAM17 (0.63) ADAM17MMP9MMP13ALDH1A1MMP1
SCHEMBL7466803 0.81 ADAM17 (0.59) ADAM17MMP9MMP13MMP1
SCHEMBL3940241 0.80 ADAM17 (0.73) ADAM17MMP9MMP13MMP1
SCHEMBL3941406 0.80 ADAM17 (0.56) ADAM17MMP9MMP13MMP1
SCHEMBL3945185 0.79 ADAM17 (0.59) ADAM17MMP9MMP13MMP1
SCHEMBL6789274 0.78 MAPT (0.44) ADAM17MMP9MMP13MAPTL3MBTL1
SCHEMBL7418210 0.78 ADAM17 (0.57) ADAM17MMP9MMP13MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147080-A1 ALKYNYL CONTAINING HYDROXAMIC ACID COMPOUNDS AS TACE INHIBITORS American Cyanamid Company (US) 2001-10-24 EP claimed
WO-2000044713-A1 ALKYNYL CONTAINING HYDROXAMIC ACID COMPOUNDS AS TACE INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-08-03 WO claimed
EP-1147080-A1 ALKYNYL CONTAINING HYDROXAMIC ACID COMPOUNDS AS TACE INHIBITORS American Cyanamid Company (US) 2001-10-24 EP disclosed
WO-2000044713-A1 ALKYNYL CONTAINING HYDROXAMIC ACID COMPOUNDS AS TACE INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-08-03 WO disclosed