SCHEMBL7415353

SCHEMBL7415353

N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)CCc1ccccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.41
CYP2D6 P10635 2/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
CYP3A4 P08684 1/20 0.41
PTPRA P18433 1/20 0.40
HRH1 P35367 2/20 0.40
KMT2A Q03164 1/20 0.39
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PPARG P37231 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415350 1.00 CYP1A2 (0.41) CYP1A2CYP2D6MAPTTSHRSMN1; SMN2
SCHEMBL7418519 0.83 SLC15A1 (0.42)
SCHEMBL7418523 0.83 SLC15A1 (0.42)
SCHEMBL27345872 0.74 SLC15A1 (0.44) CYP2D6
SCHEMBL8853856 0.73 ALDH1A1 (0.38) CYP1A2CYP2D6MAPTTSHRSMN1; SMN2
SCHEMBL10622532 0.72 EPHX1 (0.48) CYP2D6
SCHEMBL6556276 0.72 EPHX1 (0.48) CYP2D6
SCHEMBL6894985 0.72 CYP1A2 (0.55) CYP1A2CYP2D6MAPTTSHRSMN1; SMN2
SCHEMBL3348729 0.72 CYP1A2 (0.55) CYP1A2CYP2D6MAPTTSHRSMN1; SMN2
Hydrochloric Acid SCHEMBL5711578 0.71 EPHX1 (0.47) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5256677-A Enzyme inhibitor for treating acquired immune deficiency syndrome ABBOTT LABORATORIES (US) 1993-10-26 US disclosed
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO disclosed
US-5151438-A Enzyme inhibitors for treatment of aids ABBOTT LABORATORIES (US) 1992-09-29 US disclosed