SCHEMBL7415366

SCHEMBL7415366

O=C(c1cccc(C(F)(F)F)c1)C1CCN(Cc2ccccc2)C1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.66
OPRM1 P35372 1/20 0.66
OPRD1 P41143 1/20 0.66
MEN1 O00255 2/20 0.64
KMT2A Q03164 2/20 0.64
CCR2 P41597 1/20 0.62
GAA P10253 1/20 0.59
ALDH1A1 P00352 2/20 0.59
S1PR5 Q9H228 2/20 0.57
S1PR1 P21453 1/20 0.57
GRK5 P34947 1/20 0.57
CDK8 P49336 1/20 0.57
SIGMAR1 Q99720 1/20 0.57
LMNA P02545 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
NPSR1 Q6W5P4 1/20 0.55
UBE2M P61081 1/20 0.55
DCUN1D1 Q96GG9 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9650084 0.84 HTR2A (0.71) KDM4ESIGMAR1LMNA
SCHEMBL7416122 0.84 CYP3A4 (0.70) MEN1KMT2AALDH1A1S1PR5
Hydrochloric Acid SCHEMBL9649714 0.83 HTR2A (0.70) KDM4EOPRM1OPRD1SIGMAR1LMNA
SCHEMBL7415229 0.81 KMT2A (0.61) KDM4EOPRM1OPRD1MEN1KMT2A
SCHEMBL4000036 0.80 S1PR5 (0.58) KDM4EMEN1KMT2AGAAALDH1A1
SCHEMBL5539621 0.80 SIGMAR1 (0.65) SIGMAR1
SCHEMBL29783820 0.78 SIGMAR1 (0.67) KDM4EGAAALDH1A1S1PR5S1PR1
SCHEMBL4958680 0.78 SIGMAR1 (0.67) KDM4EGAAALDH1A1S1PR5S1PR1
SCHEMBL7418001 0.78 SLC18A3 (0.73) KDM4E
SCHEMBL11521377 0.78 LMNA (0.57) KDM4EOPRM1OPRD1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5198449-A N-substituted alpha-arylazacycloalkylmethanamines and their use as cardiovascular agents A. H. ROBINS COMPANY INCORPORATED (US) 1993-03-30 US disclosed