SCHEMBL7415423

SCHEMBL7415423

CC(=O)Nc1ccc(C(=O)NC(CC2CCCCC2)C(=O)N(C(C)C)C2(C#N)CCNCC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.43
CTSL P07711 6/20 0.43
CTSB P07858 3/20 0.43
CTSK P43235 2/20 0.43
USP30 Q70CQ3 5/20 0.41
BACE1 P56817 1/20 0.38
GRN P28799 1/20 0.34
SORT1 Q99523 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414894 0.90 CTSS (0.45) CTSSCTSLCTSBCTSKUSP30
SCHEMBL7414874 0.85 CTSS (0.46) CTSSCTSLCTSBCTSKUSP30
SCHEMBL7414674 0.80 CTSS (0.45) CTSSCTSLCTSBCTSKUSP30
SCHEMBL7410718 0.79 CTSS (0.47) CTSSCTSLCTSBCTSKUSP30
SCHEMBL7417185 0.78 CTSL (0.57) CTSSCTSLCTSBCTSKUSP30
SCHEMBL7415420 0.78 CTSS (0.50) CTSSCTSLCTSBCTSKUSP30
SCHEMBL7409657 0.77 CTSS (0.60) CTSSCTSLCTSBCTSKUSP30
SCHEMBL7013440 0.74 CTSL (0.40) CTSSCTSLCTSBCTSK
SCHEMBL5359753 0.74 CTSL (0.63) CTSSCTSLCTSBCTSKUSP30
SCHEMBL7014338 0.73 CTSS (0.44) CTSSCTSLCTSBCTSKUSP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed