SCHEMBL7416413

SCHEMBL7416413

COc1ccc(C(CC(=O)O)NC(=O)[C@H](CC(C)C)N2C(=O)N(Cc3ccc(NC(=O)Nc4ccccc4)cc3)C3(CCCCC3)C2=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.40
ITGA4 P13612 1/20 0.40
ITGB7 P26010 1/20 0.40
HIF1A Q16665 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HTT P42858 1/20 0.37
FPR1 P21462 2/20 0.37
FPR2 P25090 2/20 0.37
ANPEP P15144 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7105287 1.00 ITGB1 (0.40) ITGB1ITGA4ITGB7HIF1ANPC1
Tromethamine SCHEMBL7100487 0.95 ITGB1 (0.37) ITGB1ITGA4ITGB7HIF1ANPC1
SCHEMBL7101545 0.95 ITGB1 (0.48) ITGB1ITGA4ITGB7
SCHEMBL7416547 0.95 ITGB1 (0.48) ITGB1ITGA4ITGB7
SCHEMBL7107550 0.94 LMNA (0.37) ITGB1ITGA4NPC1RAB9AALDH1A1
SCHEMBL1820746 0.94 LMNA (0.37) ITGB1ITGA4NPC1RAB9AALDH1A1
SCHEMBL7100997 0.93 HIF1A (0.40) HIF1ANPC1RAB9AANPEPALDH1A1
SCHEMBL7103777 0.93 LMNA (0.37) ITGB1ITGA4NPC1RAB9APOLB
SCHEMBL1825542 0.91 ITGB1 (0.42) ITGB1ITGA4ALDH1A1MAPTHPGD
SCHEMBL7384383 0.91 ITGB1 (0.42) ITGB1ITGA4ALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183241-A1 SPIROIMIDAZOLIDINE DERIVATIVES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL PREPARATIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2002-03-06 EP disclosed
WO-2000069831-A1 SPIROIMIDAZOLIDINE DERIVATIVES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL PREPARATIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-11-23 WO disclosed