SCHEMBL7416481

SCHEMBL7416481

N#Cc1cccc(CN2CC[C@H](NC(=O)c3cccc([N+](=O)[O-])c3)C2=O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.45
KMT2A Q03164 2/20 0.45
ALDH1A1 P00352 3/20 0.43
KCNH2 Q12809 2/20 0.43
KCNJ1 P48048 1/20 0.43
POLB P06746 2/20 0.42
CCR2 P41597 1/20 0.42
ACKR3 P25106 1/20 0.41
RORC P51449 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HPGD P15428 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
CYP3A4 P08684 1/20 0.40
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
PGGT1B P53609 1/20 0.40
CHRM3 P20309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420601 0.92 KCNH2 (0.48) BRD4KMT2AALDH1A1KCNH2KCNJ1
SCHEMBL7424674 0.87 HDAC1 (0.52) BRD4KCNH2ACKR3CYP3A4FNTA
SCHEMBL7421293 0.86 BRD4 (0.47) BRD4KCNH2ACKR3RORCCYP3A4
SCHEMBL7428971 0.85 BRD4 (0.48) BRD4KMT2AALDH1A1KCNH2ACKR3
SCHEMBL7423020 0.85 CCR3 (0.46) BRD4KMT2AKCNH2ACKR3RORC
SCHEMBL7421559 0.85 F10 (0.56)
SCHEMBL7420641 0.84 BRD4 (0.43) BRD4KCNH2KCNJ1CYP3A4FNTA
SCHEMBL7419869 0.84 MCHR1 (0.49) BRD4KMT2AALDH1A1CHRM3MEN1
SCHEMBL7416484 0.83 FNTA (0.50) KMT2AALDH1A1KCNH2KCNJ1POLB
SCHEMBL7418733 0.83 CCKBR (0.52) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853618-A4 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2000-03-15 EP disclosed
EP-0853618-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1998-07-22 EP disclosed
WO-1996040679-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHÔNE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-12-19 WO disclosed