SCHEMBL7420641

SCHEMBL7420641

N#Cc1cccc(CN2CC[C@H](NC(=O)c3ccccc3[N+](=O)[O-])C2=O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.43
HSD11B1 P28845 1/20 0.43
FNTA P49354 5/20 0.42
FNTB P49356 5/20 0.42
PGGT1B P53609 5/20 0.42
KCNH2 Q12809 3/20 0.42
CYP3A4 P08684 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
PTGER4 P35408 1/20 0.40
FAAH O00519 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
RIPK1 Q13546 1/20 0.39
HTT P42858 1/20 0.39
KCNJ1 P48048 1/20 0.39
CTSD P07339 1/20 0.38
CCR3 P51677 1/20 0.38
NPY1R P25929 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420601 0.85 KCNH2 (0.48) BRD4HSD11B1FNTAFNTBPGGT1B
SCHEMBL7420645 0.84 FNTA (0.49) FNTAFNTBPGGT1BKCNH2CYP3A4
SCHEMBL7416481 0.84 BRD4 (0.45) BRD4FNTAFNTBPGGT1BKCNH2
SCHEMBL7425743 0.83 F10 (0.56)
SCHEMBL7424674 0.83 HDAC1 (0.52) BRD4FNTAFNTBPGGT1BKCNH2
SCHEMBL7425776 0.83 CCR3 (0.45) BRD4HSD11B1RIPK1CCR3
SCHEMBL7423007 0.79 GRM5 (0.52) FNTAFNTBPGGT1BKCNH2CYP3A4
SCHEMBL7418733 0.79 CCKBR (0.52) BRD4HDAC1HDAC8HDAC6
SCHEMBL7420184 0.79 SRC (0.49) BRD4HSD11B1FNTAFNTBPGGT1B
SCHEMBL7417098 0.79 ROCK2 (0.47) BRD4HSD11B1FNTAFNTBPGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853618-A4 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2000-03-15 EP disclosed
EP-0853618-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1998-07-22 EP disclosed
WO-1996040679-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHÔNE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-12-19 WO disclosed