SCHEMBL7416672

SCHEMBL7416672

COc1ccc2c(c1)C(C1(CC(C)C)CCC1)=NCC2

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.39
ALDH1A1 P00352 3/20 0.37
LMNA P02545 2/20 0.37
KDM4E B2RXH2 2/20 0.37
CYP19A1 P11511 3/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
CYP3A4 P08684 1/20 0.36
POLA1 P09884 2/20 0.36
CYP11B2 P19099 2/20 0.35
MAPT P10636 1/20 0.34
MPI P34949 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
EHMT2 Q96KQ7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747277 0.75 NPY5R (0.43) MAOAALDH1A1KDM4ECYP19A1MAPT
SCHEMBL12629538 0.74 MAPT (0.41) MAOAALDH1A1LMNAKDM4ECYP19A1
SCHEMBL989046 0.73 SLC6A2 (0.47) MAOAALDH1A1KDM4EMAPTMPI
SCHEMBL7475657 0.71 NPY5R (0.43) MAOAALDH1A1KDM4ECYP19A1CYP11B2
SCHEMBL989662 0.70 SLC6A2 (0.49) ALDH1A1LMNAKDM4ECYP19A1CYP11B2
SCHEMBL1862319 0.70 KDM4E (0.36) MAOAALDH1A1KDM4EPOLA1MAPT
SCHEMBL17375509 0.69 ALDH1A1 (0.51) MAOAALDH1A1LMNAKDM4ECYP19A1
SCHEMBL8747341 0.69 MAPK14 (0.40) MAOAALDH1A1LMNAMAPTCA1
SCHEMBL1010356 0.69 MAOA (0.60) MAOAALDH1A1LMNAKDM4ECYP19A1
SCHEMBL29664763 0.69 MAOA (0.60) MAOAALDH1A1LMNAKDM4ECYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807868-A ANALGESICS; PSYCHOLOGICAL DISORDES; PARKINSON*S DIESASE;COGNITION ACTIVATORS; DRUG DEPENDENCE; DYSKINESIA KNOLL AKTIENGESELLSCHAFT (DE) 1998-09-15 US disclosed
US-5804586-A ANALGESICS, PSYCHOLOGICAL DISORDERS KNOLL AKTIENGESELLSCHAFT (DE) 1998-09-08 US disclosed
EP-0707570-B1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1998-05-06 EP disclosed
EP-0707570-A1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS Knoll AG (DE) 1996-04-24 EP disclosed
WO-1995000489-A1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-01-05 WO disclosed