SCHEMBL7416684

SCHEMBL7416684

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2c(F)cccc2F)C(=O)O)cc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.52
ITGA2B P08514 19/20 0.52
ITGB1 P05556 1/20 0.44
ITGA5 P08648 1/20 0.44
ITGAV P06756 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7412989 0.96 ITGB3 (0.48) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7422891 0.90 ITGB3 (0.53) ITGB3ITGA2B
SCHEMBL7418686 0.89 ITGB1 (0.51) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7412996 0.87 ITGB3 (0.39) ITGB3ITGA2BITGB1ITGA5ITGAV
Trifluoroacetic Acid SCHEMBL7414096 0.86 ITGB3 (0.50) ITGB3ITGA2B
Trifluoroacetic Acid SCHEMBL7415321 0.86 ITGB1 (0.49) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7414099 0.86 ITGB3 (0.53) ITGB3ITGA2BITGAV
SCHEMBL7409585 0.86 ITGB3 (0.61) ITGB3ITGA2BITGAV
SCHEMBL7415995 0.86 ITGB3 (0.51) ITGB3ITGA2BITGAV
SCHEMBL7696995 0.85 ITGB3 (0.53) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US claimed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP claimed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO claimed