SCHEMBL7418686

SCHEMBL7418686

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2c(Cl)cccc2Cl)C(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 6/20 0.51
ITGA5 P08648 6/20 0.51
ITGB3 P05106 11/20 0.49
ITGA2B P08514 10/20 0.49
LMNA P02545 1/20 0.45
PKM P14618 1/20 0.45
ITGAV P06756 2/20 0.44
PPARG P37231 1/20 0.43
SLC1A3 P43003 1/20 0.42
SLC1A2 P43004 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7415321 0.95 ITGB1 (0.49) ITGB1ITGA5ITGB3ITGA2BLMNA
SCHEMBL7423110 0.94 ITGB3 (0.48) ITGB1ITGA5ITGB3ITGA2BLMNA
SCHEMBL7419721 0.91 ITGB3 (0.48) ITGB1ITGA5ITGB3ITGA2BITGAV
Trifluoroacetic Acid SCHEMBL7408417 0.91 ITGB1 (0.47) ITGB1ITGA5ITGB3ITGA2BLMNA
SCHEMBL7421304 0.90 ITGB3 (0.49) ITGB1ITGA5ITGB3ITGA2BITGAV
SCHEMBL7409546 0.90 ITGB3 (0.51) ITGB1ITGA5ITGB3ITGA2BITGAV
SCHEMBL7416684 0.89 ITGB3 (0.52) ITGB1ITGA5ITGB3ITGA2BITGAV
SCHEMBL7700410 0.88 ITGB3 (0.50) ITGB1ITGA5ITGB3ITGA2BITGAV
Trifluoroacetic Acid SCHEMBL7415214 0.87 ITGB3 (0.45) ITGB1ITGA5ITGB3ITGA2BITGAV
SCHEMBL7463784 0.86 ITGB3 (0.48) ITGB1ITGA5ITGB3ITGA2BITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US claimed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP claimed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO claimed