SCHEMBL7416744

SCHEMBL7416744

O=C1c2c(c3ccccc3[nH]c2=O)C(=O)N1c1ccccn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
HPGD P15428 3/20 0.47
LMNA P02545 2/20 0.47
GAA P10253 2/20 0.47
MAPK1 P28482 1/20 0.47
FGFR1 P11362 1/20 0.44
FLT1 P17948 1/20 0.44
MAPK14 Q16539 2/20 0.44
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
PADI4 Q9UM07 3/20 0.43
TNKS O95271 1/20 0.42
CYP1A2 P05177 1/20 0.42
GPR3 P46089 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42
PARP15 Q460N3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7409290 0.79 MAPK14 (0.53) PARP1SMN1; SMN2MEN1KMT2AHPGD
SCHEMBL7415475 0.78 MAPT (0.49) PARP1SMN1; SMN2MEN1KMT2AHPGD
SCHEMBL7414758 0.76 HTT (0.54) PARP1GAAMAPK1MAPK14KDM4E
SCHEMBL7415108 0.73 CASP3 (0.55) PARP1MEN1KMT2ALMNAFGFR1
SCHEMBL7406002 0.73 MAPK14 (0.44) PARP1MEN1KMT2ALMNAMAPK14
SCHEMBL7412697 0.73 ADORA3 (0.51) PARP1SMN1; SMN2MEN1KMT2ALMNA
SCHEMBL7407990 0.73 MAPK14 (0.53) PARP1MEN1KMT2ALMNAGAA
SCHEMBL7412708 0.72 CDK5 (0.43) PARP1SMN1; SMN2MEN1KMT2AHPGD
SCHEMBL7415495 0.71 KDM4E (0.40) PARP1SMN1; SMN2MEN1KMT2AHPGD
SCHEMBL30566301 0.71 SMN1; SMN2 (0.61) SMN1; SMN2MEN1KMT2AHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994026741-A1 CERTAIN PYRROLOQUINOLINONES; A NEW CLASS OF GABE BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1994-11-24 WO claimed
US-5243049-A Gamma-aminobutyric acid antagonist NEUROGEN CORPORATION (US) 1993-09-07 US claimed
US-5908932-A Certain pyrroloquinolinones; a new class of GABA brain receptor NEUROGEN CORPORATION (US) 1999-06-01 US disclosed
US-5604235-A DIAGNOSIS AND TREATMENT OF ANXIETY, SLEEP AND SEIZURE DISORDERS, BENZODIAZEPINE OVERDOSE; ENHANCEMENT OF MEMORY NEUROGEN CORPORATION (US) 1997-02-18 US disclosed
WO-1994026741-A1 CERTAIN PYRROLOQUINOLINONES; A NEW CLASS OF GABE BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1994-11-24 WO disclosed
US-5243049-A Gamma-aminobutyric acid antagonist NEUROGEN CORPORATION (US) 1993-09-07 US disclosed