SCHEMBL7416858

SCHEMBL7416858

N#Cc1cc(CN2CC[C@H](N)C2=O)co1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.33
TNKS O95271 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MAPT P10636 1/20 0.32
APEX1 P27695 1/20 0.32
F10 P00742 1/20 0.32
FNTA P49354 3/20 0.30
FNTB P49356 3/20 0.30
PGGT1B P53609 3/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423394 1.00 DPP4 (0.33) DPP4TNKSTNKS2CYP3A4TSHR
SCHEMBL7416855 0.83 SIRT2 (0.34) TNKSTNKS2F10
SCHEMBL8040069 0.75 TNKS (0.41) DPP4TNKSTNKS2CYP3A4FNTA
SCHEMBL7424938 0.75 FNTA (0.47) DPP4CYP3A4FNTAFNTBPGGT1B
SCHEMBL7418123 0.75 CHRM2 (0.35) DPP4CYP3A4TSHRTDP1MAPT
SCHEMBL7417093 0.75 CHRM2 (0.35) DPP4CYP3A4TSHRTDP1MAPT
Hydrochloric Acid SCHEMBL2328814 0.74 FNTA (0.47) DPP4CYP3A4FNTAFNTBPGGT1B
Hydrochloric Acid SCHEMBL2328817 0.74 FNTA (0.47) DPP4CYP3A4FNTAFNTBPGGT1B
SCHEMBL7422788 0.74 TRPA1 (0.36) TNKSTNKS2CYP3A4TSHRTDP1
SCHEMBL7416243 0.74 TRPA1 (0.36) TNKSTNKS2CYP3A4TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853618-A4 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2000-03-15 EP disclosed
EP-0853618-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1998-07-22 EP disclosed
WO-1996040679-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHÔNE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-12-19 WO disclosed