SCHEMBL7417331

SCHEMBL7417331

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2cccc(Cl)c2Cl)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 5/20 0.40
ITGA5 P08648 5/20 0.40
ITGB3 P05106 5/20 0.38
ITGAV P06756 4/20 0.38
ITGA2B P08514 3/20 0.36
F2 P00734 5/20 0.34
TMPRSS6 Q8IU80 4/20 0.34
POLB P06746 1/20 0.34
PPARG P37231 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415119 0.94 ITGB1 (0.39) ITGB1ITGA5ITGB3ITGAVITGA2B
SCHEMBL7416127 0.93 ITGB3 (0.37) ITGB1ITGA5ITGB3ITGA2BF2
SCHEMBL7414443 0.92 ITGB1 (0.39) ITGB1ITGA5ITGB3ITGAVITGA2B
SCHEMBL7415327 0.91 ITGB1 (0.42) ITGB1ITGA5ITGB3ITGAVITGA2B
Trifluoroacetic Acid SCHEMBL7417323 0.90 ITGB1 (0.47) ITGB1ITGA5ITGB3ITGAVITGA2B
SCHEMBL7414232 0.89 ITGB3 (0.37) ITGB1ITGA5ITGB3ITGA2BF2
SCHEMBL7408422 0.88 ITGB1 (0.40) ITGB1ITGA5ITGB3ITGAVITGA2B
SCHEMBL7694227 0.88 F10 (0.41) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7414101 0.88 ITGB3 (0.40) ITGB3ITGA2BF2TMPRSS6POLB
SCHEMBL7416348 0.87 ITGB3 (0.36) ITGB1ITGA5ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed