SCHEMBL7414101

SCHEMBL7414101

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2ccccc2F)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.40
ITGA2B P08514 11/20 0.40
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
F2 P00734 4/20 0.38
TMPRSS6 Q8IU80 4/20 0.38
POLB P06746 1/20 0.38
KAT6A Q92794 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415119 0.91 ITGB1 (0.39) ITGB3ITGA2BALDH1A1F2TMPRSS6
SCHEMBL7413080 0.91 MMP7 (0.40) ITGB3ITGA2BF2TMPRSS6POLB
SCHEMBL7415446 0.91 ITGB3 (0.39) ITGB3ITGA2BF2TMPRSS6POLB
SCHEMBL7414402 0.91 POLB (0.49) ITGB3ITGA2BF2TMPRSS6POLB
SCHEMBL7412996 0.91 ITGB3 (0.39) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7694227 0.90 F10 (0.41) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7415041 0.90 AR (0.38) ITGB3ITGA2BF2TMPRSS6POLB
SCHEMBL7417592 0.89 ITGB3 (0.49) ITGB3ITGA2BF2TMPRSS6
Trifluoroacetic Acid SCHEMBL7414096 0.89 ITGB3 (0.50) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7415626 0.89 HRH2 (0.37) ITGB3ITGA2BF2TMPRSS6POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed