SCHEMBL7417447

SCHEMBL7417447

Cc1c(C(C)C)ccc2[nH]c(N3CCCNCC3)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.45
TLR9 Q9NR96 3/20 0.44
TLR8 Q9NR97 3/20 0.44
TLR7 Q9NYK1 3/20 0.44
HTR3A P46098 2/20 0.43
NCF1 P14598 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
PRKCI P41743 1/20 0.35
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
HTR2A P28223 1/20 0.34
HTR7 P34969 1/20 0.34
HTR2B P41595 1/20 0.34
HTR6 P50406 1/20 0.34
PARP1 P09874 1/20 0.34
ROCK2 O75116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414570 0.74 HTR3A (0.40) PIM1HTR3APARP1
SCHEMBL7600366 0.71 HTR3A (0.59) PIM1HTR3AHRH4BCHEACHE
SCHEMBL13894488 0.69 NPC1 (0.65) HTR3ABCHEACHE
SCHEMBL20458912 0.69 HTR3A (0.44) PIM1TLR9TLR8HTR3APARP1
SCHEMBL3075702 0.68 HTR3A (0.88) PIM1HTR3ANCF1BCHEACHE
SCHEMBL18930378 0.68 HSD17B10 (0.41) HTR3APARP1
SCHEMBL7415578 0.68 PIM1 (0.40) PIM1HTR3AHRH4HRH3PARP1
SCHEMBL5621907 0.68 PARP1 (0.66) PARP1
Bromide SCHEMBL6599072 0.67 HTR3A (0.85) PIM1HTR3ANCF1BCHEACHE
SCHEMBL7463681 0.67 ADRB1 (0.44) PIM1HTR3AHRH4BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed