SCHEMBL7414570

SCHEMBL7414570

CC(C)c1ccc2[nH]c(N3CCNCC3)nc2c1OC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.40
PARP1 P09874 9/20 0.35
ITGB3 P05106 3/20 0.35
ITGA2B P08514 3/20 0.35
NAMPT P43490 1/20 0.35
PIM1 P11309 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410717 0.75 PARP1 (0.39) PARP1
SCHEMBL7417447 0.74 PIM1 (0.45) HTR3APARP1PIM1
SCHEMBL7417446 0.74 HTR3A (0.40) HTR3APARP1ITGB3ITGA2BNAMPT
SCHEMBL7415905 0.74 PARP1 (0.50) PARP1
SCHEMBL20458912 0.73 HTR3A (0.44) HTR3APARP1ITGB3ITGA2BNAMPT
SCHEMBL7411210 0.72 PARP1 (0.37) PARP1
SCHEMBL7409889 0.72 PARP1 (0.50) PARP1PIM1
SCHEMBL7415578 0.71 PIM1 (0.40) HTR3APARP1ITGB3ITGA2BPIM1
SCHEMBL20449682 0.69 PARP1 (0.56) HTR3APARP1KDM4E
SCHEMBL17697629 0.68 CRBN (0.59) HTR3APARP1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed