SCHEMBL7417641

SCHEMBL7417641

O=[C]c1cc(Br)c2ccccc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.43
GRM5 P41594 1/20 0.43
GRM2 Q14416 2/20 0.39
KMT2A Q03164 3/20 0.38
C1R P00736 2/20 0.38
BACE1 P56817 2/20 0.38
KDM4E B2RXH2 4/20 0.37
ALDH1A1 P00352 4/20 0.37
HPGD P15428 3/20 0.36
MAOA P21397 2/20 0.36
GLA P06280 2/20 0.36
CASP1 P29466 2/20 0.36
CASP7 P55210 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HSD17B10 Q99714 2/20 0.36
CHRM2 P08172 1/20 0.36
ADRA2A P08913 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
CHRM1 P11229 1/20 0.36
NQO2 P16083 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18585567 0.81 KDM4E (0.50) KCNH2GRM5GRM2KMT2ABACE1
SCHEMBL7666919 0.78 MYC (0.44) KCNH2KMT2AKDM4EALDH1A1HPGD
SCHEMBL3085385 0.78 CYP1A2 (0.58) KMT2ABACE1KDM4EALDH1A1HPGD
SCHEMBL7024735 0.76 ACACA (0.46) GRM2KMT2AKDM4EALDH1A1HPGD
SCHEMBL1257332 0.74 BACE1 (0.44) KCNH2GRM2KMT2AC1RBACE1
SCHEMBL7259981 0.74 ACHE (0.47) KCNH2KMT2ABACE1KDM4EALDH1A1
SCHEMBL29726892 0.74 BACE1 (0.44) KCNH2GRM2KMT2AC1RBACE1
SCHEMBL5679983 0.74 ALOX15 (0.58) KCNH2GRM5KMT2AC1RKDM4E
SCHEMBL7417644 0.72 KDM4E (0.45) KCNH2GRM2KMT2AC1RBACE1
SCHEMBL25330955 0.71 NQO2 (0.43) KCNH2GRM2KMT2ABACE1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013066-A1 CYCLIC AMIDES OF 3-AMINO-2-HYDROXY-CARBOXYLIC ACIDS AS HIV-PROTEASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1993-07-08 WO disclosed