SCHEMBL7417866

SCHEMBL7417866

[N]c1ccc([N+](=O)[O-])c2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.61
CTSB P07858 5/20 0.60
ALDH1A1 P00352 5/20 0.53
AR P10275 1/20 0.50
HSD17B10 Q99714 2/20 0.46
HPRT1 P00492 1/20 0.46
CYP3A4 P08684 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
CASP6 P55212 2/20 0.42
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
GAA P10253 1/20 0.42
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
BRD4 O60885 1/20 0.42
LMNA P02545 1/20 0.42
HSP90AA1 P07900 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7788656 0.87 TDP1 (0.80) TDP1CTSBALDH1A1ARHSD17B10
SCHEMBL57166 0.77 TDP1 (1.00) TDP1CTSBALDH1A1HSD17B10CYP3A4
SCHEMBL29475175 0.77 TDP1 (1.00) TDP1CTSBALDH1A1HSD17B10CYP3A4
SCHEMBL6815901 0.75 TDP1 (0.61) TDP1CTSBALDH1A1ARHSD17B10
SCHEMBL297029 0.75 TDP1 (0.61) TDP1CTSBALDH1A1ARHSD17B10
SCHEMBL3606794 0.75 TDP1 (0.61) TDP1CTSBALDH1A1ARHSD17B10
SCHEMBL589663 0.75 CTSB (1.00) TDP1CTSBALDH1A1ARCYP3A4
SCHEMBL16990730 0.75 TDP1 (0.61) TDP1CTSBALDH1A1ARHSD17B10
SCHEMBL8722948 0.75 TDP1 (0.61) TDP1CTSBALDH1A1ARHSD17B10
SCHEMBL1379532 0.75 TDP1 (0.61) TDP1CTSBALDH1A1ARHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773411-A CARDIOVASCULAR DISORDERS AND BRAIN DISORDERS AND COAGULANTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-06-30 US disclosed
EP-0672059-A1 CYCLIC COMPOUNDS LINKED BY A HETEROCYCLIC RING USEFUL AS INHIBITORS OF PLATELET GLYCOPROTEIN IIb/IIIa THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-09-20 EP disclosed
WO-1994011398-A1 CYCLIC COMPOUNDS LINKED BY A HETEROCYCLIC RING USEFUL AS INHIBITORS OF PLATELET GLYCOPROTEIN IIb/IIIa THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-05-26 WO disclosed