SCHEMBL7418317

SCHEMBL7418317

NC(=O)C1CC(O)CCN1C(=O)[CH]Cc1nc2ccccc2s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
HPGD P15428 3/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
LTA4H P09960 4/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
KCNH2 Q12809 1/20 0.38
MAPT P10636 2/20 0.37
UBE2T Q9NPD8 1/20 0.37
ASIC3 Q9UHC3 1/20 0.37
USP30 Q70CQ3 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ALOX15 P16050 1/20 0.37
HTT P42858 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7443421 0.87 NPC1 (0.40) ALDH1A1HPGDKMT2AMEN1LTA4H
SCHEMBL7434422 0.87 ALDH1A1 (0.39) ALDH1A1HPGDKMT2AMEN1LTA4H
SCHEMBL7359248 0.87 ALDH1A1 (0.39) ALDH1A1HPGDKMT2AMEN1LTA4H
SCHEMBL7422678 0.86 ALDH1A1 (0.38) ALDH1A1HPGDKMT2AMEN1LTA4H
SCHEMBL7420793 0.84 ALDH1A1 (0.36) ALDH1A1HPGDKMT2AMEN1LTA4H
SCHEMBL7448927 0.79 DRD2 (0.40) ALDH1A1HPGDKMT2AMEN1LTA4H
SCHEMBL3133531 0.78 DPP4 (0.38) ALDH1A1RAB9ANPC1SMN1; SMN2CYP2C19
SCHEMBL7426597 0.76 DRD2 (0.39) ALDH1A1HPGDKMT2AMEN1LTA4H
SCHEMBL6052882 0.76 SCN3A (0.41) ALDH1A1KCNH2
SCHEMBL6165827 0.75 LMNA (0.42) KMT2AMEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815103-A1 TRYPSIN AND THROMBIN INHIBITORS Novartis AG (CH) 1998-01-07 EP disclosed
WO-1996029327-A1 TRYPSIN AND THROMBIN INHIBITORS NOVARTIS AG (CH) 1996-09-26 WO disclosed