SCHEMBL7418327

SCHEMBL7418327

COc1cc2c(cc1C)CCNC2(OC(=O)C(=O)OC1(C2(c3ccsc3)CC2)NCCc2cc(C)c(OC)cc21)C1(c2ccsc2)CC1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 4/20 0.33
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL7418326 0.67 PKM (0.43) MEN1KMT2A
SCHEMBL7417327 0.65 PKM (0.46) MEN1KMT2A
SCHEMBL7411591 0.60 MAOA (0.41)
SCHEMBL8546801 0.60 POLA1 (0.38) KMT2A
SCHEMBL7411687 0.59 MAOA (0.40) MEN1KMT2A
SCHEMBL6086554 0.58 RXRA (0.46)
SCHEMBL3548729 0.58 ABCB1 (0.36)
SCHEMBL4654263 0.58 RXRA (0.37)
SCHEMBL3546929 0.57 HCRTR1 (0.40) MEN1KMT2A
SCHEMBL7417209 0.57 NAMPT (0.47) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807868-A ANALGESICS; PSYCHOLOGICAL DISORDES; PARKINSON*S DIESASE;COGNITION ACTIVATORS; DRUG DEPENDENCE; DYSKINESIA KNOLL AKTIENGESELLSCHAFT (DE) 1998-09-15 US disclosed
US-5804586-A ANALGESICS, PSYCHOLOGICAL DISORDERS KNOLL AKTIENGESELLSCHAFT (DE) 1998-09-08 US disclosed
EP-0707570-B1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1998-05-06 EP disclosed
EP-0707570-A1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS Knoll AG (DE) 1996-04-24 EP disclosed
WO-1995000489-A1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-01-05 WO disclosed