SCHEMBL7423110

SCHEMBL7423110

Cc1cccc(Cl)c1S(=O)(=O)N[C@@H](Cc1ccc(OCCCONC(=N)N)cc1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 12/20 0.48
ITGA2B P08514 9/20 0.48
ITGB1 P05556 4/20 0.48
ITGA5 P08648 4/20 0.48
ITGAV P06756 3/20 0.45
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
PPARG P37231 2/20 0.42
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7408417 0.96 ITGB1 (0.47) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7418686 0.94 ITGB1 (0.51) ITGB3ITGA2BITGB1ITGA5ITGAV
Trifluoroacetic Acid SCHEMBL7415321 0.90 ITGB1 (0.49) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7700410 0.89 ITGB3 (0.50) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7463784 0.89 ITGB3 (0.48) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7414099 0.87 ITGB3 (0.53) ITGB3ITGA2BITGAVPPARGMMP2
SCHEMBL7408422 0.87 ITGB1 (0.40) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7421304 0.86 ITGB3 (0.49) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7409546 0.86 ITGB3 (0.51) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7418575 0.86 ITGB3 (0.55) ITGB3ITGA2BITGB1ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US claimed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP claimed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO claimed