SCHEMBL7418948

SCHEMBL7418948

NC(=O)C(N)NC(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 0.47
ICAM1 P05362 1/20 0.47
ITGAL P20701 1/20 0.47
ALDH1A1 P00352 3/20 0.44
JAK2 O60674 2/20 0.44
TYK2 P29597 2/20 0.44
HPGD P15428 1/20 0.44
CYP3A4 P08684 1/20 0.44
JAK1 P23458 1/20 0.44
KMT2A Q03164 1/20 0.43
MAPT P10636 2/20 0.42
PPIA P62937 1/20 0.41
GAA P10253 2/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
TAS1R2 Q8TE23 1/20 0.41
KDM4E B2RXH2 1/20 0.41
APAF1 O14727 1/20 0.41
TDP2 O95551 1/20 0.41
NSD2 O96028 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8804032 0.81 ITGB2 (0.46) ITGB2ICAM1ITGALALDH1A1JAK2
SCHEMBL7411826 0.81 ITGB2 (0.46) ITGB2ICAM1ITGALALDH1A1JAK2
SCHEMBL7417230 0.80 ITGB2 (0.43) ITGB2ICAM1ITGALALDH1A1JAK2
SCHEMBL7419439 0.77 ITGB2 (0.43) ITGB2ICAM1ITGALALDH1A1JAK2
SCHEMBL11056940 0.76 ALDH1A1 (0.49) ALDH1A1JAK2TYK2HPGDCYP3A4
SCHEMBL7411327 0.75 ITGB2 (0.44) ITGB2ICAM1ITGALALDH1A1JAK2
Water SCHEMBL7924276 0.74 TAS1R3 (0.47) ALDH1A1JAK2TYK2HPGDCYP3A4
SCHEMBL7418492 0.73 ITGB2 (0.43) ITGB2ICAM1ITGALALDH1A1JAK2
SCHEMBL11440641 0.73 JAK2 (0.53) ALDH1A1JAK2TYK2HPGDCYP3A4
SCHEMBL4377125 0.72 ALDH1A1 (0.56) ALDH1A1JAK2TYK2HPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157003-A1 ACYLATED AMINOACETONITRILES AS CYSTEINE PROTEASE INHIBITORS AstraZeneca AB (SE) 2001-11-28 EP disclosed
WO-2000048992-A1 ACYLATED AMINOACETONITRILES AS CYSTEINE PROTEASE INHIBITORS ASTRAZENECA AB (SE) 2000-08-24 WO disclosed