SCHEMBL7411327

SCHEMBL7411327

CC(NC(=O)c1c(Cl)cccc1Cl)C(N)=S

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 0.44
ICAM1 P05362 1/20 0.44
ITGAL P20701 1/20 0.44
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
TYK2 P29597 3/20 0.41
ALDH1A1 P00352 2/20 0.41
JAK2 O60674 2/20 0.41
HPGD P15428 1/20 0.41
CYP3A4 P08684 1/20 0.41
JAK1 P23458 1/20 0.41
ITGB1 P05556 3/20 0.40
ITGA4 P13612 3/20 0.40
KMT2A Q03164 1/20 0.40
PSMB5 P28074 1/20 0.40
TAS1R3 Q7RTX0 2/20 0.39
TAS1R1 Q7RTX1 2/20 0.39
TAS1R2 Q8TE23 2/20 0.39
RAB9A P51151 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8804032 0.87 ITGB2 (0.46) ITGB2ICAM1ITGALCTSSCTSK
SCHEMBL12020093 0.82 MAPT (0.48) CTSSCTSKALDH1A1HPGDITGB1
SCHEMBL14500982 0.81 PYGL (0.49) ITGB2ICAM1ITGALITGB1ITGA4
SCHEMBL7410618 0.80 ITGB2 (0.50) ITGB2ICAM1ITGALALDH1A1HPGD
SCHEMBL11056940 0.79 ALDH1A1 (0.49) TYK2ALDH1A1JAK2HPGDCYP3A4
Water SCHEMBL7924276 0.78 TAS1R3 (0.47) TYK2ALDH1A1JAK2HPGDCYP3A4
SCHEMBL23355170 0.76 TYK2 (0.45) ITGB2ICAM1ITGALTYK2ALDH1A1
SCHEMBL7418948 0.75 ITGB2 (0.47) ITGB2ICAM1ITGALTYK2ALDH1A1
SCHEMBL20387787 0.73 PKM (0.54) ALDH1A1HPGDITGB1ITGA4KMT2A
SCHEMBL7411826 0.73 ITGB2 (0.46) ITGB2ICAM1ITGALTYK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157003-A1 ACYLATED AMINOACETONITRILES AS CYSTEINE PROTEASE INHIBITORS AstraZeneca AB (SE) 2001-11-28 EP disclosed
WO-2000048992-A1 ACYLATED AMINOACETONITRILES AS CYSTEINE PROTEASE INHIBITORS ASTRAZENECA AB (SE) 2000-08-24 WO disclosed