SCHEMBL7419101

SCHEMBL7419101

N#CC1(N(Cc2ccccc2)C(=O)C2(NC(=O)OCc3ccccc3)CCCCC2)CCNC1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 8/20 0.53
CTSL P07711 7/20 0.53
CTSB P07858 7/20 0.53
CTSK P43235 7/20 0.43
TLR2 O60603 2/20 0.37
PREP P48147 2/20 0.35
TACR1 P25103 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7023323 0.88 CTSS (0.42) CTSSCTSLCTSBCTSK
SCHEMBL6565010 0.78 CTSS (0.34) CTSSCTSLCTSBCTSK
SCHEMBL7021490 0.76 CTSK (0.56) CTSSCTSLCTSBCTSK
SCHEMBL6184079 0.75 CTSS (0.67) CTSSCTSLCTSBCTSKTACR1
SCHEMBL7021496 0.75 CTSS (0.41) CTSSCTSLCTSBCTSK
SCHEMBL25198329 0.74 CTSS (0.50) CTSSCTSLCTSBCTSKTLR2
SCHEMBL25198330 0.74 CTSS (0.50) CTSSCTSLCTSBCTSKTLR2
SCHEMBL6183576 0.74 CTSS (0.65) CTSSCTSLCTSBCTSKPREP
SCHEMBL9900827 0.73 CTSL (0.63) CTSSCTSLCTSBCTSKPREP
SCHEMBL6567042 0.72 CTSS (0.35) CTSSCTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed