SCHEMBL6565010

SCHEMBL6565010

N#CC1(N(Cc2ccccc2)C(=O)C2(OC(=O)NCc3ccccc3)CCCCC2)CCNC1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.34
CTSB P07858 2/20 0.34
CTSL P07711 1/20 0.34
LMNA P02545 2/20 0.32
EPHX1 P07099 2/20 0.32
HPGD P15428 1/20 0.32
MCL1 Q07820 1/20 0.32
CTSK P43235 1/20 0.32
MC4R P32245 1/20 0.32
ATM Q13315 1/20 0.32
JAK3 P52333 1/20 0.32
PLIN1 O60240 1/20 0.31
PLIN5 Q00G26 1/20 0.31
ABHD5 Q8WTS1 1/20 0.31
BCHE P06276 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6567042 0.94 CTSS (0.35) CTSSCTSBCTSLLMNAEPHX1
SCHEMBL6565456 0.89 ACHE (0.38) CTSSCTSBCTSLLMNAEPHX1
SCHEMBL7431174 0.85 LMNA (0.37) CTSSCTSBCTSLLMNAEPHX1
SCHEMBL6565861 0.85 CTSB (0.36) CTSSCTSBCTSLLMNACTSK
SCHEMBL7434373 0.84 CTSB (0.40) CTSSCTSBCTSLEPHX1HPGD
SCHEMBL7419101 0.78 CTSS (0.53) CTSSCTSBCTSLCTSK
SCHEMBL7023323 0.77 CTSS (0.42) CTSSCTSBCTSLCTSK
SCHEMBL6565853 0.76 CTSL (0.42) CTSSCTSBCTSLCTSK
SCHEMBL3898232 0.75 CTSB (0.43) CTSSCTSBCTSLEPHX1HPGD
SCHEMBL6565858 0.75 NR1H4 (0.36) CTSSCTSBCTSLCTSKATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed