SCHEMBL7419310

SCHEMBL7419310

C[C@H](CO)c1ccccc1NC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.45
NLRP3 Q96P20 1/20 0.45
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
BRD9 Q9H8M2 1/20 0.40
ELANE P08246 2/20 0.40
CTRB1 P17538 1/20 0.40
METAP1 P53582 1/20 0.39
BRD4 O60885 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28514442 0.86 IDO1 (0.44) IDO1NLRP3TP53MAPTLMNA
SCHEMBL28905847 0.86 BRD9 (0.44) IDO1NLRP3TP53MAPTLMNA
SCHEMBL2737224 0.85 NLRP3 (0.56) IDO1NLRP3TP53MAPTLMNA
SCHEMBL1771858 0.84 IDO1 (0.47) IDO1NLRP3TP53MAPTLMNA
SCHEMBL17230179 0.82 IDO1 (0.44) IDO1NLRP3TP53MAPTLMNA
SCHEMBL30850148 0.81 IDO1 (0.42) IDO1NLRP3TP53MAPTLMNA
SCHEMBL24166675 0.81 IDO1 (0.43) IDO1NLRP3TP53MAPTLMNA
SCHEMBL8837511 0.81 CXCL8 (0.49) IDO1NLRP3TP53MAPTLMNA
SCHEMBL8214432 0.81 IDO1 (0.43) IDO1NLRP3TP53MAPTLMNA
SCHEMBL1951665 0.81 CXCL8 (0.49) IDO1NLRP3TP53MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0349570-A1 RENIN INHIBITORS CONTAINING A CYCLOPROPYL AMINO ACID AND/OR A CYCLOALKYL TRANSITION-STATE ANALOGUE THE UPJOHN COMPANY (US) 1990-01-10 EP disclosed
WO-1988007053-A1 RENIN INHIBITORS CONTAINING A CYCLOPROPYL AMINO ACID AND/OR A CYCLOALKYL TRANSITION-STATE ANALOGUE THE UPJOHN COMPANY (US) 1988-09-22 WO disclosed