SCHEMBL7419740

SCHEMBL7419740

C=C(C(=O)OCC)C1CCc2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 5/20 0.51
ALDH1A1 P00352 4/20 0.46
MAPT P10636 2/20 0.46
KCNQ2 O43526 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
FFAR1 O14842 2/20 0.39
PPIB P23284 1/20 0.39
PPIA P62937 1/20 0.39
XBP1 P17861 1/20 0.39
HTT P42858 1/20 0.39
ANO1 Q5XXA6 2/20 0.38
MTNR1A P48039 2/20 0.38
MTNR1B P49286 2/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720088 0.82 PIN1 (0.52) PIN1ALDH1A1MAPTFFAR1XBP1
SCHEMBL8301042 0.82 PIN1 (0.47) PIN1ALDH1A1MAPTKCNQ2L3MBTL1
SCHEMBL6781189 0.82 SRD5A1 (0.38) PIN1ALDH1A1MAPT
SCHEMBL19985038 0.81 PIN1 (0.46) PIN1ALDH1A1MAPTKCNQ2L3MBTL1
SCHEMBL23934507 0.77 ALDH1A1 (0.43) ALDH1A1MAPTL3MBTL1CA1CA2
SCHEMBL8160821 0.77 PIN1 (0.58) PIN1KCNQ2PPIBPPIAHTT
SCHEMBL19207927 0.76 PIN1 (0.42) PIN1ALDH1A1KCNQ2ANO1MTNR1A
SCHEMBL19207928 0.76 PIN1 (0.42) PIN1ALDH1A1KCNQ2ANO1MTNR1A
SCHEMBL19224562 0.76 PIN1 (0.42) PIN1ALDH1A1KCNQ2ANO1MTNR1A
SCHEMBL30327597 0.76 PIN1 (0.56) PIN1KCNQ2PPIBPPIAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5801274-A N- mercaptoacyl(amino acid or peptide)! compounds and S-lipophilic aliphatic carbonyl derivatives thereof as antihypertensives INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 1998-09-01 US disclosed
EP-0609310-B1 N-(MERCAPTOACYL)AMINO ACIDS, METHODS OF THEIR PREPARATION AND THERAPEUTIC USE, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM INST NAT SANTE RECH MED (FR) 1998-07-29 EP disclosed
US-5591891-A PEPTIDASE INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1997-01-07 US disclosed
EP-0609310-A1 N-(MERCAPTOACYL)AMINO ACIDS, METHODS OF THEIR PREPARATION AND THERAPEUTIC USE, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1994-08-10 EP disclosed
WO-1994017036-A1 S-LIPOPHILIC ALIPHATIC CARBONYL [N-MERCAPTOACYL-(AMINO ACID OR PEPTIDE)] COMPOUNDS AS ANTIHYPERTENSIVE AGENTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1994-08-04 WO disclosed
EP-0539848-A1 N-(mercaptoacyl)amino acids, methods of their preparation and therapeutic use, and pharmaceutical compositions containing them INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1993-05-05 EP disclosed
WO-1993008162-A1 N-(MERCAPTOACYL)AMINO ACIDS, METHODS OF THEIR PREPARATION AND THERAPEUTIC USE, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1993-04-29 WO disclosed