SCHEMBL7420016

SCHEMBL7420016

CNc1ccc(C2(C(=O)C3CCCC3)CC2)cc1NC(=O)CNc1ccc(C#N)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
PKM P14618 1/20 0.42
PAX8 Q06710 1/20 0.39
GAA P10253 3/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
MCHR1 Q99705 4/20 0.38
EPHX1 P07099 1/20 0.38
FASN P49327 1/20 0.36
TSHR P16473 1/20 0.35
NAMPT P43490 1/20 0.34
PGR P06401 2/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
NPC1 O15118 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7412573 0.84 ALDH1A1 (0.42) ALDH1A1PKMGAAKMT2AMAPT
SCHEMBL7409714 0.78 ALDH1A1 (0.39) ALDH1A1PKMGAAKMT2AMAPT
SCHEMBL7414201 0.75 ALDH1A1 (0.35) ALDH1A1PKMPAX8GAAKMT2A
SCHEMBL7420019 0.73 FASN (0.34) PAX8EPHX1FASNPGR
SCHEMBL7412219 0.71 F2 (0.55) ALDH1A1PKMKMT2AMEN1NPC1
SCHEMBL7412365 0.70 PRKCI (0.42) ALDH1A1GAAKMT2A
SCHEMBL7410714 0.67 HCAR3 (0.47) ALDH1A1GAAKMT2AMAPT
SCHEMBL16208436 0.65 ALDH1A1 (0.59) ALDH1A1PKMGAAKMT2AMAPT
SCHEMBL7420806 0.65 ALDH1A1 (0.38) ALDH1A1PKMGAAKMT2AMAPT
SCHEMBL28279381 0.64 ALDH1A1 (0.55) ALDH1A1PKMGAAKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-B1 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA (DE) 2002-12-11 EP disclosed
US-6248770-B1 CARDIOVASCULAR DISORDERS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-06-19 US disclosed
EP-0869791-A4 4-SUBSTITUTED PIPERIDINE ANALOGS AND THEIR USE AS SUBTYPE SELECTIVE NMDA RECEPTOR ANTAGONISTS WARNER LAMBERT CO (US) 1999-04-28 EP disclosed
EP-0869791-A1 4-SUBSTITUTED PIPERIDINE ANALOGS AND THEIR USE AS SUBTYPE SELECTIVE NMDA RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1998-10-14 EP disclosed
WO-1997023214-A1 4-SUBSTITUTED PIPERIDINE ANALOGS AND THEIR USE AS SUBTYPE SELECTIVE NMDA RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1997-07-03 WO disclosed