SCHEMBL7414201

SCHEMBL7414201

CCOC(=O)CCC(=O)N(C1CCCC1)C1(c2ccc(NC)c(NC(=O)CNc3ccc(C#N)cc3)c2)CC1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.35
MAPT P10636 5/20 0.35
GAA P10253 5/20 0.35
PKM P14618 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
PAX8 Q06710 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MCHR1 Q99705 1/20 0.33
MAPK1 P28482 1/20 0.33
PGR P06401 1/20 0.32
TDP1 Q9NUW8 4/20 0.32
L3MBTL1 Q9Y468 2/20 0.31
FASN P49327 3/20 0.31
CYP2D6 P10635 1/20 0.31
OPRK1 P41145 1/20 0.31
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27553886 0.85 FASN (0.34) FASN
SCHEMBL7414205 0.79 F2 (0.31) PGR
SCHEMBL7413025 0.76 F2 (0.43) MEN1KMT2ASMN1; SMN2
SCHEMBL7449396 0.76 MAPT (0.37) ALDH1A1MAPTKMT2AMAPK1FASN
SCHEMBL7420016 0.75 ALDH1A1 (0.42) ALDH1A1MAPTGAAPKMHSP90AA1
SCHEMBL7412466 0.74 MAPT (0.42) ALDH1A1MAPTGAAPKMMEN1
SCHEMBL7414208 0.73 CYP11B2 (0.33) MCHR1L3MBTL1
SCHEMBL7412573 0.70 ALDH1A1 (0.42) ALDH1A1MAPTGAAPKMMEN1
SCHEMBL7449392 0.70 NPC1 (0.34) ALDH1A1MAPTPAX8MAPK1LMNA
SCHEMBL7413022 0.69 F2 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-B1 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA (DE) 2002-12-11 EP disclosed
US-6248770-B1 CARDIOVASCULAR DISORDERS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-06-19 US disclosed
EP-1095025-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-05-02 EP disclosed
WO-2000001704-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-01-13 WO disclosed