SCHEMBL7420539

SCHEMBL7420539

CCOC(=O)[C@@H](O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CC(N)=O)NC(=O)OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PSMB1 P20618 1/20 0.55
ADORA3 P0DMS8 1/20 0.52
ADORA2A P29274 1/20 0.52
ADORA2B P29275 1/20 0.52
ADORA1 P30542 1/20 0.52
CTSL P07711 8/20 0.51
CTSB P07858 4/20 0.51
REN P00797 2/20 0.47
CTSK P43235 3/20 0.47
CTSS P25774 2/20 0.47
MME P08473 1/20 0.46
ECE1 P42892 1/20 0.46
PSMB8 P28062 1/20 0.46
PSMB5 P28074 1/20 0.46
CASP3 P42574 1/20 0.45
CASP7 P55210 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7418250 0.88 PSMB1 (0.61) PSMB1ADORA3ADORA2AADORA2BADORA1
SCHEMBL7420596 0.88 PSMB1 (0.61) PSMB1ADORA3ADORA2AADORA2BADORA1
SCHEMBL7412449 0.88 PSMB1 (0.61) PSMB1ADORA3ADORA2AADORA2BADORA1
SCHEMBL7417704 0.86 PSMB1 (0.60) PSMB1ADORA3ADORA2AADORA2BADORA1
SCHEMBL7384058 0.86 PSMB1 (0.60) PSMB1ADORA3ADORA2AADORA2BADORA1
SCHEMBL7270223 0.84 PSMB1 (0.59) PSMB1ADORA3ADORA2AADORA2BADORA1
SCHEMBL5344617 0.81 ADORA3 (0.59) PSMB1ADORA3ADORA2AADORA2BADORA1
SCHEMBL7742845 0.80 PSMB1 (0.56) PSMB1CTSLCTSBCTSKCTSS
SCHEMBL7742003 0.80 PSMB1 (0.56) PSMB1CTSLCTSBCTSKCTSS
SCHEMBL7279478 0.80 ADORA3 (0.56) PSMB1ADORA3ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013066-A1 CYCLIC AMIDES OF 3-AMINO-2-HYDROXY-CARBOXYLIC ACIDS AS HIV-PROTEASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1993-07-08 WO disclosed