SCHEMBL7420982

SCHEMBL7420982

CC(C)(C)CC(NC(=O)c1ccc(NS(C)(=O)=O)cc1)C(=O)N(Cc1ccccc1)C1(C#N)CCNC1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSL P07711 10/20 0.36
CTSS P25774 8/20 0.36
CTSK P43235 7/20 0.36
CTSB P07858 5/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ADRB1 P08588 2/20 0.35
NR3C2 P08235 1/20 0.34
EPHX2 P34913 1/20 0.34
NR1H4 Q96RI1 1/20 0.34
CTSF Q9UBX1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7419241 0.91 CTSL (0.43) CTSLCTSSCTSKCTSBKDM4E
SCHEMBL7014338 0.87 CTSS (0.44) CTSLCTSSCTSKCTSBALDH1A1
SCHEMBL7420985 0.80 ALDH1A1 (0.43) KDM4EALDH1A1ADRB1NR3C2EPHX2
SCHEMBL7014342 0.80 CTSS (0.41) CTSSKDM4EALDH1A1ADRB1EPHX2
SCHEMBL7414895 0.79 CTSL (0.47) CTSLCTSS
SCHEMBL7423676 0.75 CTSL (0.44) CTSLCTSSCTSKCTSBCTSF
SCHEMBL7419135 0.74 CTSS (0.45) CTSLCTSSCTSKCTSB
SCHEMBL7013440 0.71 CTSL (0.40) CTSLCTSSCTSKCTSBALDH1A1
SCHEMBL7414874 0.71 CTSS (0.46) CTSLCTSSCTSKCTSB
SCHEMBL7021242 0.71 CTSL (0.39) CTSLCTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed