SCHEMBL7419241

SCHEMBL7419241

CC(C)(C)CC(NC(=O)c1ccccc1)C(=O)N(Cc1ccccc1)C1(C#N)CCNC1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSL P07711 13/20 0.43
CTSS P25774 8/20 0.43
CTSB P07858 8/20 0.43
CTSK P43235 7/20 0.43
RAB9A P51151 1/20 0.39
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ATM Q13315 1/20 0.37
PTPN1 P18031 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420982 0.91 CTSL (0.36) CTSLCTSSCTSBCTSKKDM4E
SCHEMBL7414895 0.86 CTSL (0.47) CTSLCTSS
SCHEMBL7423676 0.83 CTSL (0.44) CTSLCTSSCTSBCTSKRAB9A
SCHEMBL7419135 0.79 CTSS (0.45) CTSLCTSSCTSBCTSK
SCHEMBL7419245 0.77 SIGMAR1 (0.41) CTSLCTSSCTSBCTSKRAB9A
SCHEMBL7014338 0.77 CTSS (0.44) CTSLCTSSCTSBCTSKALDH1A1
SCHEMBL7422431 0.76 CTSS (0.47) CTSLCTSSCTSBCTSKALDH1A1
SCHEMBL7021490 0.76 CTSK (0.56) CTSLCTSSCTSBCTSK
SCHEMBL7021242 0.75 CTSL (0.39) CTSLCTSSCTSBCTSK
SCHEMBL7417228 0.74 CTSL (0.44) CTSLCTSSCTSBCTSKATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed