SCHEMBL7422260

SCHEMBL7422260

N#Cc1c(Cl)cccc1Oc1ccc(S(=O)(=O)N[C@@H](Cc2ccc(OCCCONC(=N)N)cc2)C(=O)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.48
BCL2L1 Q07817 1/20 0.45
MCL1 Q07820 1/20 0.45
ITGB3 P05106 5/20 0.44
ITGA2B P08514 5/20 0.44
HSD11B1 P28845 1/20 0.44
MMP2 P08253 7/20 0.43
MMP9 P14780 5/20 0.43
ITGB1 P05556 1/20 0.42
ITGA5 P08648 1/20 0.42
ADAMTS5 Q9UNA0 1/20 0.41
KCNA5 P22460 1/20 0.41
MMP3 P08254 1/20 0.40
MMP13 P45452 1/20 0.40
ADAMTS4 O75173 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7413027 0.96 MAPT (0.45) MAPTBCL2L1MCL1ITGB3ITGA2B
SCHEMBL7413033 0.89 MAPT (0.41) MAPTBCL2L1MCL1ITGB3ITGA2B
SCHEMBL7417646 0.83 MMP2 (0.56) ITGB3ITGA2BMMP2MMP9ADAMTS5
SCHEMBL7418686 0.82 ITGB1 (0.51) ITGB3ITGA2BITGB1ITGA5
SCHEMBL7463648 0.82 MAPT (0.46) MAPTBCL2L1MCL1ITGB3ITGA2B
SCHEMBL7409585 0.82 ITGB3 (0.61) ITGB3ITGA2BMMP2MMP9KCNA5
SCHEMBL7409554 0.81 MMP2 (0.61) ITGB3ITGA2BMMP2MMP9ADAMTS5
SCHEMBL7696995 0.81 ITGB3 (0.53) ITGB3ITGA2BMMP2MMP9KCNA5
SCHEMBL7419820 0.80 ITGB3 (0.48) ITGB3ITGA2BMMP2MMP9ITGB1
SCHEMBL7420817 0.80 ITGB3 (0.56) ITGB3ITGA2BMMP2MMP9KCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US claimed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP claimed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO claimed