SCHEMBL7422355

SCHEMBL7422355

CCOC(=O)C(CN[C@@H](CC(C)C)C(=O)OCc1ccccc1)c1ccc(-c2ccncc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.44
MAPT P10636 4/20 0.42
NPSR1 Q6W5P4 2/20 0.42
CTSK P43235 8/20 0.42
CTSL P07711 5/20 0.42
HSD17B10 Q99714 1/20 0.41
CTSS P25774 5/20 0.41
CTSB P07858 3/20 0.41
ALDH1A1 P00352 2/20 0.41
NTSR1 P30989 1/20 0.41
ATM Q13315 1/20 0.41
RECQL P46063 1/20 0.41
S1PR4 O95977 1/20 0.40
S1PR1 P21453 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420936 0.92 CTSL (0.41) MAPTNPSR1CTSKCTSLHSD17B10
SCHEMBL7415848 0.91 CTSK (0.45) MAPTNPSR1CTSKCTSLHSD17B10
SCHEMBL7429552 0.88 HSD17B10 (0.45) MAPTNPSR1CTSKCTSLHSD17B10
SCHEMBL7426033 0.88 MAPT (0.42) MAPTNPSR1CTSKCTSLHSD17B10
SCHEMBL7421323 0.84 NTSR1 (0.44) AAK1MAPTNPSR1CTSKCTSL
SCHEMBL5870517 0.81 AAK1 (0.46) AAK1CTSKCTSLHSD17B10
SCHEMBL5870515 0.81 AAK1 (0.46) AAK1CTSKCTSLHSD17B10
SCHEMBL5870522 0.81 AAK1 (0.46) AAK1CTSKCTSLHSD17B10
SCHEMBL27300721 0.79 HSD17B10 (0.48) MAPTNPSR1CTSKCTSLHSD17B10
SCHEMBL18775038 0.79 CTSK (0.56) MAPTCTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed