SCHEMBL7422377

SCHEMBL7422377

NC(=O)/C1=C/C=C\Cc2ccccc2O1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
ATM Q13315 1/20 0.34
NOTUM Q6P988 2/20 0.34
TRPA1 O75762 2/20 0.33
PARP1 P09874 4/20 0.32
HSD17B3 P37058 1/20 0.32
ALOX5 P09917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9319857 0.85 MAOA (0.38) MAOAMAOBNOTUMHSD17B3ALOX5
SCHEMBL29569443 0.81 MAOA (0.41) MAOAMAOBATMNOTUMTRPA1
SCHEMBL2971412 0.81 MAOA (0.41) MAOAMAOBATMNOTUMTRPA1
Hydrochloric Acid SCHEMBL19744197 0.80 MAOA (0.39) MAOAMAOBATMNOTUMTRPA1
SCHEMBL11551370 0.79 MAOA (0.38) MAOAMAOB
SCHEMBL11556597 0.76 MAOA (0.42) MAOAMAOBATM
Trifluoroacetic Acid SCHEMBL29570875 0.73 MAOA (0.33) MAOAMAOBATMNOTUMTRPA1
SCHEMBL5848189 0.73 TRPA1 (0.41) ATMTRPA1PARP1
SCHEMBL9259332 0.71 MAOA (0.41) MAOAMAOBATM
Acetamide SCHEMBL7696552 0.70 SMN1; SMN2 (0.38) MAOAMAOBATMNOTUMPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5288731-A Antiemetics, antiserotonine agents RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1994-02-22 US disclosed
WO-1992009284-A1 2,6-METHANO-2H-1-BENZOXOCINCARBOXAMIDES AS 5-HT3-ANTAGONISTS RHONE-POULENC RORER INTERNATIONAL (HOLDINGS), INC. (US) 1992-06-11 WO disclosed