SCHEMBL7422898

SCHEMBL7422898

O=c1[nH]nc2c3ccccc3ncn12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.55
HPGD P15428 1/20 0.55
HSD17B10 Q99714 1/20 0.55
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
LTK P29376 2/20 0.43
ALK Q9UM73 2/20 0.43
DYRK1B Q9Y463 2/20 0.43
RET P07949 1/20 0.43
MET P08581 1/20 0.43
GRK5 P34947 1/20 0.43
CDK8 P49336 1/20 0.43
RPS6KA3 P51812 1/20 0.43
MST1R Q04912 1/20 0.43
TYRO3 Q06418 1/20 0.43
DYRK1A Q13627 1/20 0.43
LRRK2 Q5S007 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
SMN1; SMN2 Q16637 4/20 0.42
RAB9A P51151 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420880 0.80 KDM4E (0.47) KDM4EHPGDHSD17B10SMN1; SMN2RAB9A
SCHEMBL18229915 0.78 PDE3B (0.49) KDM4EHPGDHSD17B10PDE3BPDE3A
SCHEMBL3479430 0.78 LTK (0.41) PDE3BPDE3ALTKALKDYRK1B
SCHEMBL30759507 0.78 PDE3B (0.49) KDM4EHPGDHSD17B10PDE3BPDE3A
SCHEMBL30636803 0.71 KDM4E (1.00) KDM4EHPGDHSD17B10SMN1; SMN2RAB9A
SCHEMBL10969790 0.71 KDM4E (0.57) KDM4EHPGDHSD17B10SMN1; SMN2RAB9A
SCHEMBL2119422 0.71 LTK (0.51) HSD17B10PDE3BPDE3ALTKALK
SCHEMBL4787828 0.71 KDM4E (1.00) KDM4EHPGDHSD17B10SMN1; SMN2RAB9A
SCHEMBL4517379 0.70 PDE5A (0.49) HSD17B10PDE3BPDE3ALTKALK
SCHEMBL30434733 0.69 PDE5A (0.55) KDM4EHPGDPDE3BPDE3ALTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999018106-A1 NOVEL 1,2,4-TRIAZOLO[4,3-C]QUINAZOLIN-3-ONES AND 1,2,4-TRIAZOLO[4,3-C]QUINAZOLIN-3-THIONES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1999-04-15 WO disclosed
WO-1999018106-A1 NOVEL 1,2,4-TRIAZOLO[4,3-C]QUINAZOLIN-3-ONES AND 1,2,4-TRIAZOLO[4,3-C]QUINAZOLIN-3-THIONES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1999-04-15 WO disclosed
US-4463007-A ANTIALLERGENS BASF AKTIENGESELLSCHAFT (DE) 1984-07-31 US disclosed