SCHEMBL7423210

SCHEMBL7423210

CCOC(=O)CN(c1ccc(N)cc1)S(=O)(=O)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.55
NR1I2 O75469 1/20 0.55
MAPK1 P28482 2/20 0.50
USP2 O75604 2/20 0.50
KEAP1 Q14145 2/20 0.50
NFE2L2 Q16236 2/20 0.50
HCRTR2 O43614 4/20 0.49
TSHR P16473 1/20 0.48
NR3C1 P04150 1/20 0.48
LMNA P02545 1/20 0.47
PTPN1 P18031 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5479473 0.86 HCRTR2 (0.52) ALDH1A1NR1I2MAPK1USP2KEAP1
SCHEMBL7422328 0.83 KMT2A (0.64) ALDH1A1NR1I2MAPK1KEAP1NFE2L2
SCHEMBL6318614 0.82 ALDH1A1 (0.48) ALDH1A1USP2TSHRLMNAPTPN1
SCHEMBL5624368 0.82 LMNA (0.45) ALDH1A1HCRTR2TSHRLMNAPTPN1
SCHEMBL3462930 0.82 HCRTR2 (0.53) ALDH1A1NR1I2MAPK1KEAP1NFE2L2
SCHEMBL6573645 0.81 KEAP1 (0.48) ALDH1A1KEAP1NFE2L2HCRTR2
SCHEMBL7000752 0.81 KEAP1 (0.66) ALDH1A1MAPK1KEAP1NFE2L2LMNA
SCHEMBL7003143 0.79 KEAP1 (0.71) ALDH1A1KEAP1NFE2L2HCRTR2LMNA
SCHEMBL1732616 0.78 SMN1; SMN2 (0.49) ALDH1A1MAPK1USP2HCRTR2TSHR
SCHEMBL27599056 0.78 SMN1; SMN2 (0.49) ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885205-A4 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2002-11-27 EP disclosed
EP-0885205-A1 FIBRINOGEN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-12-23 EP disclosed
US-5780480-A THROMBOLYTIC AGENTS, ANTICOAGULANTS MERCK & CO., INC. (US) 1998-07-14 US disclosed
WO-1997031910-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-09-04 WO disclosed